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机构 日期 题名 作者
臺大學術典藏 2022-05-12T03:49:29Z Identification of Entry Inhibitors against Delta and Omicron Variants of SARS-CoV-2 Lee, Richard Kuan-Lin; Li, Tian-Neng; SUI-YUAN CHANG; Chao, Tai-Ling; Kuo, Chun-Hsien; Pan, Max Yu-Chen; Chiou, Yu-Ting; Liao, Kuan-Ju; Yang, Yi; Wu, Yi-Hsuan; Huang, Chen-Hao; Juan, Hsueh-Fen; Hsieh, Hsing-Pang; Wang, Lily Hui-Ching
臺大學術典藏 2022-04-14T23:27:22Z Identification of Entry Inhibitors against Delta and Omicron Variants of SARS-CoV-2 Lee, Richard Kuan Lin; Li, Tian Neng; SUI-YUAN CHANG; Chao, Tai Ling; Kuo, Chun Hsien; Pan, Max Yu Chen; Chiou, Yu Ting; Liao, Kuan Ju; Yang, Yi; Wu, Yi Hsuan; Huang, Chen Hao; HSUEH-FEN JUAN; Hsieh, Hsing Pang; Wang, Lily Hui Ching
國立交通大學 2019-04-02T06:00:35Z Structural Basis for the Improved Potency of Peroxisome Proliferator-Activated Receptor (PPAR) Agonists Peng, Yi-Hui; Coumar, Mohane Selvaraj; Leou, Jiun-Shyang; Wu, Jian-Sung; Shiao, Hui-Yi; Lin, Chia-Hui; Lin, Wen-Hsing; Lien, Tzu Wen; Chen, Xin; Hsu, John T. -A.; Chao, Yu-Sheng; Huang, Chien-Fu; Lyu, Ping-Chiang; Hsieh, Hsing-Pang; Wu, Su-Ying
國立交通大學 2019-04-02T06:00:18Z Design and Synthesis of Tetrahydropyridothieno[2,3-d]pyrimidine Scaffold Based Epidermal Growth Factor Receptor (EGFR) Kinase Inhibitors: The Role of Side Chain Chirality and Michael Acceptor Group for Maximal Potency Wu, Chia-Hsien; Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Wen-Hsing; Chen, Yi-Rong; Chen, Chiung-Tong; Shiao, Hui-Yi; Rafi, Shaik; Wang, Sing-Yi; Hsu, Hui; Chen, Chun-Hwa; Chang, Chun-Yu; Chang, Teng-Yuan; Lien, Tzu-Wen; Fang, Ming-Yu; Yeh, Kai-Chia; Chen, Ching-Ping; Yeh, Teng-Kuang; Hsieh, Su-Huei; Hsu, John T. -A.; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立成功大學 2016 Disruption of protein-protein interactions: hot spot detection, structure-based virtual screening and in vitro testing for the anti-cancer drug target survivin Sarvagalla, Sailu; Cheung, Chun Hei Antonio; Tsai, Ju-Ya; Hsieh, Hsing Pang; Coumar, Mohane Selvaraj
國立交通大學 2015-11-26T00:57:01Z 發展以DBPR104為主之抗體藥物複合體:設計、合成與藥物活性評估 李志揚; Lee, Chih-Yang; 謝興邦; 李耀坤; 許馨云; Hsieh, Hsing-Pang; Li, Yaw-Kuen; Hsu, Hsin-Yun
國立交通大學 2014-12-08T15:48:06Z Structural Basis for the Improved Potency of Peroxisome Proliferator-Activated Receptor (PPAR) Agonists Peng, Yi-Hui; Coumar, Mohane Selvaraj; Leou, Jiun-Shyang; Wu, Jian-Sung; Shiao, Hui-Yi; Lin, Chia-Hui; Lin, Wen-Hsing; Lien, Tzu Wen; Chen, Xin; Hsu, John T. -A.; Chao, Yu-Sheng; Huang, Chien-Fu; Lyu, Ping-Chiang; Hsieh, Hsing-Pang; Wu, Su-Ying
國立交通大學 2014-12-08T15:48:04Z Design and Synthesis of Tetrahydropyridothieno[2,3-d]pyrimidine Scaffold Based Epidermal Growth Factor Receptor (EGFR) Kinase Inhibitors: The Role of Side Chain Chirality and Michael Acceptor Group for Maximal Potency Wu, Chia-Hsien; Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Wen-Hsing; Chen, Yi-Rong; Chen, Chiung-Tong; Shiao, Hui-Yi; Rafi, Shaik; Wang, Sing-Yi; Hsu, Hui; Chen, Chun-Hwa; Chang, Chun-Yu; Chang, Teng-Yuan; Lien, Tzu-Wen; Fang, Ming-Yu; Yeh, Kai-Chia; Chen, Ching-Ping; Yeh, Teng-Kuang; Hsieh, Su-Huei; Hsu, John T. -A.; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:29:53Z Parallel Screening of Wild-Type and Drug-Resistant Targets for Anti-Resistance Neuraminidase Inhibitors Hsu, Kai-Cheng; Hung, Hui-Chen; Horng, Jim-Tong; Fang, Ming-Yu; Chang, Chun-Yu; Li, Ling-Ting; Chen, I-Jung; Chen, Yun-Chu; Chou, Ding-Li; Chang, Chun-Wei; Hsieh, Hsing-Pang; Yang, Jinn-Moon; Hsu, John T. -A.
國立交通大學 2014-12-08T15:21:34Z A High-throughput Cell-based Screening for L858R/T790M Mutant Epidermal Growth Factor Receptor Inhibitors Lin, Wen-Hsing; Song, Jen-Shin; Lien, Tzu-Wen; Chang, Chun-Yu; Wu, Szu-Huei; Huang, Yu-Wen; Chang, Teng-Yuan; Fang, Ming-Yu; Yen, Kuei-Jung; Chen, Chun-Hwa; Chu, Chang-Ying; Hsieh, Hsing-Pang; Chen, Yi-Rong; Chao, Yu-Sheng; Hsu, John T-A
國立交通大學 2014-12-08T15:21:24Z Identification of BPR3P0128 as an Inhibitor of Cap-Snatching Activities of Influenza Virus Hsu, John T. -A.; Yeh, Jiann-Yih; Lin, Ta-Jen; Li, Mei-ling; Wu, Ming-Sian; Hsieh, Chung-Fan; Chou, Yao Chieh; Tang, Wen-Fang; Lau, Kean Seng; Hung, Hui-Chen; Fang, Ming-Yu; Ko, Shengkai; Hsieh, Hsing-Pang; Horng, Jim-Tong
國立交通大學 2014-12-08T15:13:45Z Anti-influenza drug discovery Hsu, John T.-A.; Hsieh, Hsing-Pang; Hung, Hui-Chen; Ju, Yi Wei; Tseng, Sung-Nain; Tseng, C.-P.; Yang, Jinn-Moon; Chang, Chun-Wei; Fang, Min-Yu; Lin, Chun-Cheng; Homg, Jim-Tong; Shih, Shin-Ru; Chao, Yu-Sheng
國立交通大學 2014-12-08T15:10:01Z Aurintricarboxylic acid inhibits influenza virus neuraminidase Hung, Hui-Chen; Tseng, Ching-Ping; Yang, Jinn-Moon; Ju, Yi-Wei; Tseng, Sung-Nain; Chen, Yen-Fu; Chao, Yu-Sheng; Hsieh, Hsing-Pang; Shih, Shin-Ru; Hsu, John T. -A.
國立交通大學 2014-12-08T15:09:36Z Design and Structural Analysis of Novel Pharmacophores for Potent and Selective Peroxisome Proliferator-activated Receptor gamma Agonists Lin, Chia-Hui; Peng, Yi-Hui; Coumar, Mohane Selvaraj; Chittimalla, Santhosh Kumar; Liao, Chun-Chen; Lyn, Ping-Chiang; Huang, Chin-Chieh; Lien, Tzu-Wen; Lin, Wen-Hsing; Hsu, John T. -A.; Cheng, Jai-Hong; Chen, Xin; Wu, Jian-Sung; Chao, Yu-Sheng; Lee, Hwei-Jen; Juo, Chiun-Gung; Wu, Su-Ying; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:07:38Z BPR2-D2 targeting viral ribonucleoprotein complex-associated function inhibits oseltamivir-resistant influenza viruses Shih, Shin-Ru; Horng, Jim-Tong; Poon, Leo L. M.; Chen, Tzu-Chun; Yeh, Jiann-Yih; Hsieh, Hsing-Pang; Tseng, Sung-Nain; Chiang, Chiayn; Li, Wan-Ling; Chao, Yu-Sheng; Hsu, John T. -A.
國立交通大學 2014-12-08T15:07:27Z Identification, SAR Studies, and X-ray Co-crystallographic Analysis of a Novel Furanopyrimidine Aurora Kinase A Inhibitor Coumar, Mohane Selvaraj; Tsai, Ming-Tsung; Chu, Chang-Ying; Uang, Biing-Jiun; Lin, Wen-Hsing; Chang, Chun-Yu; Chang, Teng-Yuan; Leou, Jiun-Shyang; Teng, Chi-Huang; Wu, Jian-Sung; Fang, Ming-Yu; Chen, Chun-Hwa; Hsu, John T-A; Wu, Su-Ying; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:07:23Z Anti-Influenza Drug Discovery: Structure-Activity Relationship and Mechanistic Insight into Novel Angelicin Derivatives Yeh, Jiann-Yih; Coumar, Mohane Selvaraj; Horng, Jim-Tong; Shiao, Hui-Yi; Kuo, Fu-Ming; Lee, Hui-Ling; Chen, In-Chun; Chang, Chun-Wei; Tang, Wen-Fang; Tseng, Sung-Nain; Chen, Chi-Jene; Shih, Shin-Ru; Hsu, John T. -A; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:07:23Z Pyrazole compound BPR1P0034 with potent and selective anti-influenza virus activity Shih, Shin-Ru; Chu, Tzu-Yun; Reddy, Gadarla Randheer; Tseng, Sung-Nain; Chen, Hsiun-Ling; Tang, Wen-Fang; Wu, Ming-sian; Yeh, Jiann-Yih; Chao, Yu-Sheng; Hsu, John T. A.; Hsieh, Hsing-Pang; Horng, Jim-Tong
國立交通大學 2014-12-08T15:06:34Z Fast-Forwarding Hit to Lead: Aurora and Epidermal Growth Factor Receptor Kinase Inhibitor Lead Identification Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Cheng-Wei; Shiao, Hui-Yi; Ho, Yun-Lung; Reddy, Randheer; Lin, Wen-Hsing; Chen, Chun-Hwa; Peng, Yi-Hui; Leou, Jiun-Shyang; Lien, Tzu-Wen; Huang, Chin-Ting; Fang, Ming-Yu; Wu, Szu-Huei; Wu, Jian-Sung; Chittimalla, Santhosh Kumar; Song, Jen-Shin; Hsu, John T. -A.; Wu, Su-Ying; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立成功大學 2014-08-01 CDKN1A-mediated responsiveness of MLL-AF4-positive acute lymphoblastic leukemia to Aurora kinase-A inhibitors Chen, Ya-Ping; Lin, Hui-Ju; Chen, Jiann-Shiuh; Tsai, Ming-Ying; Hsieh, Hsing-Pang; Chang, Jang-Yang; Chen, Nai-Feng; Chang, Kung-Chao; Huang, Wen-Tsung; Su, Wu-Chou; Yang, Shu-Ting; Chang, Wen-Chang; Hung, Liang-Yi; Chen, Tsai-Yun
臺北醫學大學 2014 CDKN1A-mediated Responsiveness of MLL-AF4-positive Acute Lymphoblastic Leukemia to Aurora Kinase-A Inhibitors Chen, Ya-Ping;Lin, Hui-Ju;Chen, Jiann-Shiuh;Tsai, Ming-Ying;Hsieh, Hsing-Pang;Chang, Jang-Yang;Chen, Nai-Feng;Chang, Kung-Chao;Huang, Wen-Tsung;Su, Wu-Chou;Shu-Ti
國立成功大學 2013 Pronounced induction of endoplasmic reticulum stress and tumor suppression by surfactant-free poly(lactic-co-glycolic acid) nanoparticles via modulation of the PI3K signaling pathway Hou, Chia-Cheng; Tsai, Tsung-Lin; Su, Wen-Pin; Hsieh, Hsing-Pang; Yeh, Chen-Sheng; Shieh, Dar-Bin; Su, Wu-Chou
國立成功大學 2011-08-24 BPR1K653, a Novel Aurora Kinase Inhibitor, Exhibits Potent Anti-Proliferative Activity in MDR1 (P-gp170)-Mediated Multidrug-Resistant Cancer Cells Cheung, Chun Hei Antonio; Lin, Wen-Hsing; Hsu, John Tsu-An; Hour, Tzyh-Chyuan; Yeh, Teng-Kuang; Ko, Shengkai; Lien, Tzu-Wen; Coumar, Mohane Selvaraj; Liu, Jin-Fen; Lai, Wen-Yang; Shiao, Hui-Yi; Lee, Tian-Ren; Hsieh, Hsing-Pang; Chang, Jang-Yang
國立成功大學 2011-03-07 2-Amino-3,4,5-Trimethoxybenzophenones as Potent Tubulin Polymerization Inhibitors Chuang, Hsun-Yueh; Chang, Jang-Yang; Lai, Mei-Jung; Kuo, Ching-Chuan; Lee, Hsueh-Yun; Hsieh, Hsing-Pang; Chen, Ying-Jen; Chen, Li-Tzong; Pan, Wen-Yu; Liou, Jing-Ping
國立臺灣大學 2011 Inhibition of Hiv-1 Tat-Mediated Transcription by a Coumarin Derivative, Bprhiv001, through the Akt Pathway 林必涵; 柯屹又; 蘇峻霆; 蕭暉議; 謝興邦; 趙昱凱; 李君男; 高全良; 趙宇生; 張淑媛; LIN, PI-HAN; KE, YI-YU; SU, CHUN-TING; SHIAO, HUI-YI; HSIEH, HSING-PANG; CHAO, YU-KAI; LEE, CHUN-NAN; KAO, CHUAN-LIANG; CHAO, YU-SHENG; CHANG, SUI-YUAN
國立成功大學 2009-07-03 Survivin counteracts the therapeutic effect of microtubule de-stabilizers by stabilizing tubulin polymers Cheung, Chun Hei Antonio; Chen, Huang-Hui; Kuo, Ching-Chuan; Chang, Chi-Yen; Coumar, Mohane S.; Hsieh, Hsing-Pang; Chang, Jang-Yang
國立成功大學 2009-04 Synthesis and Structure-Activity Relationships of 1-Benzyl-4,5,6-trimethoxyindoles as a Novel Class of Potent Antimitotic Agents Lai, Mei-Jung; Kuo, Ching-Chuan; Yeh, Teng-Kuang; Hsieh, Hsing-Pang; Chen, Li-Tzong; Pan, Wen-Yu; Hsu, Kuang-Yang; Chang, Jang-Yang; Liou, Jing-Ping
國立臺灣大學 2009 Bortezomib Overcomes Trail Resistance in Hepatocellular Carcinoma Cells in Part through the Inhibition of P13k/Akt Pathway 陳昆鋒; 葉培彥; 許駿; 徐志宏; 盧彥伸; 謝興邦; 陳培哲; 鄭安理; CHEN, KUEN-FENG; YEH, PEI-YEN; HSU, CHIUN; HSU, CHIH-HUNG; LU, YEN-SHEN; HSIEH, HSING-PANG; CHEN, PEI-JER; CHENG, ANN-LII
國立臺灣大學 2009 Bortezomib Overcomes Tumor Necrosis Factor-Related Apoptosis-Inducing Ligand Resistance in Hepatocellular Carcinoma Cells in Part through the Inhibition of the Phosphatidylinositol 3-Kinase/Akt Pathway 陳昆鋒; 葉培彥; 許駿; 徐志宏; 盧彥伸; 謝興邦; 陳培哲; 鄭安理; CHEN, KUEN-FENG; YEH, PEI-YEN; HSU, CHIUN; HSU, CHIH-HUNG; LU, YEN-SHEN; HSIEH, HSING-PANG; CHEN, PEI-JER; CHENG, ANN-LII
國立成功大學 2008-12-25 Synthesis and Structure-Activity Relationships of 2-Amino-1-aroylnaphthalene and 2-Hydroxy-1-aroylnaphthalenes as Potent Antitubulin Agents Reddy, Gadarla Randheer; Kuo, Ching-Chuan; Tan, Uan-Kang; Coumar, Mullane Selvaraj; Chang, Chi-Yen; Chiang, Yi-Kun; Lai, Mei-Jung; Yeh, Jiann-Yih; Wu, Su-Ying; Chang, Jing-Yang; Liou, Jing-Ping; Hsieh, Hsing-Pang
國立成功大學 2008-07-24 Discovery of 4-amino and 4-hydroxy-1-aroylindoles as potent tubulin polymerization inhibitors Liou, Jing-Ping; Wu, Zi-Yi; Kuo, Ching-Chuan; Chang, Chi-Yen; Lu, Pei-Yi; Chen, Chi-Ming; Hsieh, Hsing-Pang; Chang, Jang-Yang
國立臺灣大學 2008 Thiopurine analogues inhibit papain-like protease of severe acute respiratory syndrome coronavirus Chou, Chi-Yuan; Chien, Chia-Hui; Han, Yu-San; Prebanda, Mojca Trstenjak; Hsieh, Hsing-Pang; Turk, Boris; Chang, Gu-Gang; Chen, Xin
國立臺灣大學 2008 Anti-Hsv Activity of Digitoxin and Its Possible Mechanisms 蘇峻霆; 徐祖安; 謝興邦; 陳廷祺; 高全良; 李君男; 張淑媛; SU, CHUN-TING; HSU, JOHN TSU-AN; HSIEH, HSING-PANG; CHEN, TING-CHI; KAO, CHUAN-LIANG; LEE, CHUN-NAN; CHANG, SUI-YUAN
國立臺灣大學 2006 Discovery of a novel family of SARS-CoV protease inhibitors by virtual screening and 3D-QSAR studies Tsai, Keng-Chang; Chen, Shih-Yuan; Liang, Po-Huang; Lu, I-Lin; Mahindroo, Neeraj; Hsieh, Hsing-Pang; Chao, Yu-Sheng; Liu, Lincoln; Liu, Donald; Lien, Wei; Lin, Thy-Hou; Wu, Su-Ying
國立臺灣大學 2006 Structure-Based Drug Design and Structural Biology Study of Novel Nonpeptide Inhibitors of Severe Acute Respiratory Syndrome Coronavirus Main Protease Lu, I-Lin; Mahindroo, Neeraj; Liang, Po-Huang; Peng, Yi-Hui; Kuo, Chih-Jung; Tsai, Keng-Chang; Hsieh, Hsing-Pang; Chao, Yu-Sheng; Wu, Su-Ying
臺大學術典藏 2006 Discovery of a novel family of SARS-CoV protease inhibitors by virtual screening and 3D-QSAR studies Tsai, Keng-Chang; Chen, Shih-Yuan; Liang, Po-Huang; Lu, I-Lin; Mahindroo, Neeraj; Hsieh, Hsing-Pang; Chao, Yu-Sheng; Liu, Lincoln; Liu, Donald; Lien, Wei; Lin, Thy-Hou; Wu, Su-Ying; Tsai, Keng-Chang; Chen, Shih-Yuan et al.
國立臺灣大學 2004 A Novel Bis-Benzylidenecyclopentanone Derivative, Bpr0y007, Inducing a Rapid Caspase Activation Involving Upregulation of Fas (Cd95/Apo-1) and Wild-Type P53 in Human Oral Epidermoid Carcinoma Cells 潘文玉; 郭靜娟; 劉景平; 洪怡玫; 陳立宗; 謝興邦; 張俊彥; PAN, WEN-YU; KUO, CHING-CHUAN; LIOU, JING-PING; HUNG, YI-MEI; CHEN, LI-TZONG; HSIEH, HSING-PANG; CHANG, JANG-YANG
國立臺灣大學 1999 Direct solid-phase synthesis of octreotide conjugates: precursors for use as tumor-targeted radiopharmaceuticals Hsieh, Hsing-Pang; Wu, Ying-Ta; Chen, Shui-Tein; Wang, Kung-Tsung
國立臺灣大學 1998 Facile solid phase synthesis of octreotide analogs using p-carboxybenzaldehyde as a novel linker to anchor Fmoc-threoninol to solid phase resins Wu, Ying-Ta; Hsieh, Hsing-Pang; Wu, Chi-Yu; Yu, Hui-Ming; Chen, Shui-Tein; Wang, Kung-Tsung

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