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机构 日期 题名 作者
臺大學術典藏 2021-03-02T05:49:30Z Design and synthesis of 3-benzylaminocoumarin-7-O-sulfamate derivatives as steroid sulfatase inhibitors Hng, Yue; Lin, Mei-Hsiang; Lin, Tzung-Sheng; Liu, I-Chen; Lin, I-Chun; Lu, Yeh-Lin; Chang, Chiao-Nien; Chiu, Pei-Fang; Tsai, Keng-Chang; MEI-JOU CHEN; Liang, Pi-Hui
臺大學術典藏 2021-01-09T09:27:08Z Design and synthesis of 3-benzylaminocoumarin-7-O-sulfamate derivatives as steroid sulfatase inhibitors Hng, Yue; Hng, Yue;Lin, Mei-Hsiang;Lin, Tzung-Sheng;Liu, I-Chen;Lin, I-Chun;Lu, Yeh-Lin;Chang, Chiao-Nien;Chiu, Pei-Fang;Tsai, Keng-Chang;Mei-Jou Chen;Pi-Hui Liang; Lin, Mei-Hsiang; Lin, Tzung-Sheng; Liu, I-Chen; Lin, I-Chun; Lu, Yeh-Lin; Chang, Chiao-Nien; Chiu, Pei-Fang; Tsai, Keng-Chang; MEI-JOU CHEN; PI-HUI LIANG
衛生福利部國家中醫藥研究所 2018-12-12T17:44:13Z Acylguanidine derivatives of zanamivir and oseltamivir: Potential orally available prodrugs against influenza viruses Hsu, Peng-Hao;Chiu, Din-Chi;Wu, Kuan-Lin;Lee, Pei-Shan;Jan, Jia-Tsrong;Cheng, Yih-Shyun E.;Tsai, Keng-Chang;Cheng, Ting-Jen;Fang, Jim-Min
衛生福利部國家中醫藥研究所 2018 Generation and characterization of avian-derived anti-human CD19 single chain fragment antibodies Tsai, Keng-Chang;Chiang, Chen-Wei;Lo, Yan-Ni;Chang, Fu-Ling;Lin, Tsai-Yu;Chang, Chang-Yu;Chen, Wang-Chuan;Lee, Yu-Ching
衛生福利部國家中醫藥研究所 2018 GSK-3 inhibition through GLP-1R allosteric activation mediates the neurogenesis promoting effect of P7C3 after cerebral ischemic/reperfusional injury in mice Wang, Yea-Hwey;Liou, Kuo-Tong;Tsai, Keng-Chang;Liu, Hui-Kang;Yang, Li-Ming;Chern, Chang-Ming;Shen, Yuh-Chiang
衛生福利部國家中醫藥研究所 2018 Interaction of S17 antibody with the functional binding region of the hepatitis B virus pre-S2 epitope Chang, Chang-Yu;Chang, Fu-Ling;Chiang, Chen-Wei;Lo, Yan-Ni;Lin, Tsai-Yu;Chen, Wang-Chuan;Tsai, Keng-Chang;Lee, Yu-Ching
衛生福利部國家中醫藥研究所 2018 New hirsutinolide-type sesquiterpenoids from Vernonia cinerea inhibit nitric oxide production in LPS-stimulated RAW264.7 cells Yang Kuo, Li-Ming;Tseng, Pei-Yi;Lin, Yu-Chi;Liaw, Chia-Ching;Zhang, Li-Jie;Tsai, Keng-Chang;Lin, Zhi-Hu;Ho, Hsiu-O;Kuo, Yao-Haur
衛生福利部國家中醫藥研究所 2018 Protein–DNA complex-guided discovery of the antibacterial lead E1 for restoring the susceptibility of Klebsiella Pneumoniae to polymyxin B by targeting the response regulator PmrA Tseng, Tien-Sheng;Tu, I-Fan;Chen, Hsiao-Ting;Lin, Lie-Chwen;Tsai, Keng-Chang;Wu, Shih-Hsiung;Chen, Chinpan
衛生福利部國家中醫藥研究所 2017 Protein disulfide isomerase a4 acts as a novel regulator of cancer growth through the procaspase pathway. Kuo, Tien-Fen;Chen, Tzung-Yan;Jiang, Si-Tse;Chen, Kai-Wei;Chiang, Yi-Ming;Hsu, Yi-Jou;Liu, Yan-Jun;Chen, Hui-Ming;Yokoyama, Kazunari;Tsai, Keng-Chang;Yeh, Hsu-Hua;Chen, Yet-Ran;Yang, Meng-Ting;Yang, Chun-Yen;Yang, Wen-Chin
衛生福利部國家中醫藥研究所 2017 Peramivir Conjugates as Orally Available Agents against Influenza H275Y Mutant. Wang, Peng-Cheng;Chiu, Din-Chi;Jan, Jia-Tsrong;Huang, Wen-I;Cheng, Ting-Jen;Tsai, Keng-Chang;Fang, Jim-Min
衛生福利部國家中醫藥研究所 2017 Peramivir analogues bearing hydrophilic side chains exhibit higher activities against H275Y mutant than wild-type influenza virus. Chiu, Din-Chi;Lin, Tzu-Chen;Huang, Wen-I;Cheng, Ting-Jen;Tsai, Keng-Chang;Fang, Jim-Min
衛生福利部國家中醫藥研究所 2017 Characterizing the structure-function relationship reveals the mode of action of a novel antimicrobial peptide, P1, from jumper ant Myrmecia pilosula. Tseng, Tien-Sheng;Tsai, Keng-Chang;Chen, Chin-Pan
衛生福利部國家中醫藥研究所 2016 Identifying N-linked glycan moiety and motifs in the cysteine-rich domain critical for N-glycosylation and intracellular trafficking of SR-AI and MARCO. Tsay, Huey-Jen; Huang, Yung-Cheng; Chen, Yi-Jen; Lee, Yun-Hao; Hsu, Shu-Meng; Tsai, Keng-Chang; Yang, Cheng-Ning; Huang, Fong-Lee; Shie, Feng-Shiun; Lee, Lin-Chien; Shiao, Young-Ji
衛生福利部國家中醫藥研究所 2016 Peramivir Phosphonate Derivatives as Influenza Neuraminidase Inhibitors. Wang, Peng-Cheng; Fang, Jim-Min; Tsai, Keng-Chang; Wang, Shi-Yun; Huang, Wen-I; Tseng, Yin-Chen; Cheng, Yih-Shyun E.; Cheng, Ting-Jen Rachel; Wong, Chi-Huey
衛生福利部國家中醫藥研究所 2016 Sarkosyl-Induced Helical Structure of an Antimicrobial Peptide GW-Q6 Plays an Essential Role in the Binding of Surface Receptor OprI in Pseudomonas aeruginosa Tseng, Tien-Sheng; Wang, Shih-Han; Chang, Ting-Wei; Wei, Hung-Mu; Wang, Yu-June; Tsai, Keng-Chang; Liao, You-Di; Chen, Chinpan
衛生福利部國家中醫藥研究所 2016 Predicting Ligand Binding Sites on Protein Surfaces by 3-Dimensional Probability Density Distributions of Interacting Atoms Jian, Jhih-Wei; Elumalai, Pavadai; Pitti, Thejkiran; Wu, Chih Yuan; Tsai, Keng-Chang; Chang, Jeng-Yih; Peng, Hung-Pin; Yang, An-Suei
衛生福利部國家中醫藥研究所 2016 Discovery of a potent cyclooxygenase-2 inhibitor, S4, through docking-based pharmacophore screening, in vivo and in vitro estimations Tseng, Tien-Sheng; Chuang, Show-Mei; Hsiao, Nai-Wan; Chen, Yi-Wen; Lee, Yu-Ching; Lin, Chi-Chen; Huang, Cheng; Tsai, Keng-Chang
衛生福利部國家中醫藥研究所 2015 Single chain antibody fragment with serine protease inhibitory property capable of neutralizing toxicity of Trimeresurus mucrosquamatus venom Lee, Yu-Ching; Chen, Wang-Chuan; Liang, Meng-Huei; Lee, Chi-Hsin; Tsai, Keng-Chang; Chiang, Jen-Ron; Chiang, Liao-Chun; Chen, Chi-Ching; Chang, Chang-Yu; Lee, Ching-Hsiao; Leu, Sy-Jye; Yang, Yi-Yuan
衛生福利部國家中醫藥研究所 2015 Differential inhibition of CYP1-catalyzed regioselective hydroxylation of estradiol by berberine and its oxidative metabolites Chang, Yu-Ping; Huang, Chiung-Chiao; Shen, Chien-Chang; Tsai, Keng-Chang; Ueng, Yune-Fang
衛生福利部國家中醫藥研究所 2015 Discovery of novel FFA4 (GPR120) receptor agonists with β-arrestin2-biased characteristics. Li, Ang; Yang, Duxiao; Zhu, Mengyuan; Tsai, Keng-chang; Xiao, Kun-hong; Yu, Xiao; Sun, Jinpeng; Du, Lupei
衛生福利部國家中醫藥研究所 2015 Comparative study between 3D-QSAR and Docking-Based Pharmacophore models for potent Plasomodium falciparum dihydroorotate dehydrogenase inhibitors Tseng, Tien-Sheng; Lee, Yu-Ching; Hsiao, Nai-Wan; Liu, Yun-Ru; Tsai, Keng-Chang
衛生福利部國家中醫藥研究所 2015 Discovery of highly potent tyrosinase inhibitor, T1, with significant anti-melanogenesis ability by zebrafish in vivo assay and computational molecular modeling. Chen, Wang-Chuan; Tseng, Tien-Sheng; Hsiao, Nai-Wan; Lin, Yun-Lian; Wen, Zhi-Hong; Tsai, Chin-Chuan; Lee, Yu-Ching; Lin, Hui-Hsiung; Tsai, Keng-Chang
衛生福利部國家中醫藥研究所 2015 Discovery of Potent Cysteine-Containing Dipeptide Inhibitors against Tyrosinase: A Comprehensive Investigation of 20×20 Dipeptides in Inhibiting Dopachrome Formation Tseng, Tien-Sheng;Tsai, Keng-Chang;Chen, Wang-Chuan;Wang, Yeng-Tseng;Lee, Yu-Ching;Lu, Chung-Kuang;Don, Ming-Jaw;Chang, Chang-Yu;Lee, Ching-Hsiao;Lin, Hui-Hsiung;Hsu, Hung-Ju;Hsiao, Nai-Wan
衛生福利部國家中醫藥研究所 2015 Engineering a nanopore with co-chaperonin function Ho, Ching-Wen; Meervelt, Veerle Van; Tsai, Keng-Chang; Temmerman, Pieter-Jan De; Mast, Jan; Maglia, Giovanni
衛生福利部國家中醫藥研究所 2015 The Effect of Oxidation on Berberine-Mediated CYP1 Inhibition: Oxidation Behavior and Metabolite-Mediated Inhibition. Lo, Sheng-Nan; Shen, Chien-Chang; Chang, Chia-Yu; Tsai, Keng-Chang; Huang, Chiung-Chiao; Wu, Tian-Shung; Ueng, Yune-Fang

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