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Showing items 1-14 of 14  (1 Page(s) Totally)
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Institution Date Title Author
國立成功大學 2020-08-15 The SMAC mimetic LCL161 is a direct ABCB1/MDR1-ATPase activity modulator and BIRC5/Survivin expression down-regulator in cancer cells 張雋曦; Cheung, Chun Hei Antonio; Chang, Yung-Chieh;Kondapuram, Sree Karani;Yang, Tsung-Han;Syed, Safiulla Basha;Cheng, Siao Muk;Lin, Tzu-Yu;Lin, Yi-Chen;Coumar, Mohane Selvaraj;Chang, Jang-Yang;Leung, Euphemia
國立成功大學 2020-07-02 BIRC5/Survivin is a novel ATG12–ATG5 conjugate interactor and an autophagy-induced DNA damage suppressor in human cancer and mouse embryonic fibroblast cells 張雋曦; Cheung, Chun Hei Antonio; Lin, Tzu-Yu;Chan, Hsiu-Han;Chen, Shang-Hung;Sarvagalla, Sailu;Chen, Pai-Sheng;Coumar, Mohane Selvaraj;Cheng, Siao Muk;Chang, Yung-Chieh;Lin, Chun-Hui;Leung, Euphemia
國立成功大學 2019-08 Cloning, expression, and purification of the recombinant pro-apoptotic dominant-negative Survivin T34A-C84A protein in Escherichia coli 張雋曦; Cheung, Chun Hei Antonio; Tsai, Shing-Ling;Chang, Yung-Chieh;Sarvagalla, Sailu;Wang, Shuying;Coumar, Mohane Selvaraj
國立交通大學 2019-04-02T06:00:35Z Structural Basis for the Improved Potency of Peroxisome Proliferator-Activated Receptor (PPAR) Agonists Peng, Yi-Hui; Coumar, Mohane Selvaraj; Leou, Jiun-Shyang; Wu, Jian-Sung; Shiao, Hui-Yi; Lin, Chia-Hui; Lin, Wen-Hsing; Lien, Tzu Wen; Chen, Xin; Hsu, John T. -A.; Chao, Yu-Sheng; Huang, Chien-Fu; Lyu, Ping-Chiang; Hsieh, Hsing-Pang; Wu, Su-Ying
國立交通大學 2019-04-02T06:00:18Z Design and Synthesis of Tetrahydropyridothieno[2,3-d]pyrimidine Scaffold Based Epidermal Growth Factor Receptor (EGFR) Kinase Inhibitors: The Role of Side Chain Chirality and Michael Acceptor Group for Maximal Potency Wu, Chia-Hsien; Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Wen-Hsing; Chen, Yi-Rong; Chen, Chiung-Tong; Shiao, Hui-Yi; Rafi, Shaik; Wang, Sing-Yi; Hsu, Hui; Chen, Chun-Hwa; Chang, Chun-Yu; Chang, Teng-Yuan; Lien, Tzu-Wen; Fang, Ming-Yu; Yeh, Kai-Chia; Chen, Ching-Ping; Yeh, Teng-Kuang; Hsieh, Su-Huei; Hsu, John T. -A.; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立成功大學 2016 Disruption of protein-protein interactions: hot spot detection, structure-based virtual screening and in vitro testing for the anti-cancer drug target survivin Sarvagalla, Sailu; Cheung, Chun Hei Antonio; Tsai, Ju-Ya; Hsieh, Hsing Pang; Coumar, Mohane Selvaraj
國立交通大學 2014-12-08T15:48:06Z Structural Basis for the Improved Potency of Peroxisome Proliferator-Activated Receptor (PPAR) Agonists Peng, Yi-Hui; Coumar, Mohane Selvaraj; Leou, Jiun-Shyang; Wu, Jian-Sung; Shiao, Hui-Yi; Lin, Chia-Hui; Lin, Wen-Hsing; Lien, Tzu Wen; Chen, Xin; Hsu, John T. -A.; Chao, Yu-Sheng; Huang, Chien-Fu; Lyu, Ping-Chiang; Hsieh, Hsing-Pang; Wu, Su-Ying
國立交通大學 2014-12-08T15:48:04Z Design and Synthesis of Tetrahydropyridothieno[2,3-d]pyrimidine Scaffold Based Epidermal Growth Factor Receptor (EGFR) Kinase Inhibitors: The Role of Side Chain Chirality and Michael Acceptor Group for Maximal Potency Wu, Chia-Hsien; Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Wen-Hsing; Chen, Yi-Rong; Chen, Chiung-Tong; Shiao, Hui-Yi; Rafi, Shaik; Wang, Sing-Yi; Hsu, Hui; Chen, Chun-Hwa; Chang, Chun-Yu; Chang, Teng-Yuan; Lien, Tzu-Wen; Fang, Ming-Yu; Yeh, Kai-Chia; Chen, Ching-Ping; Yeh, Teng-Kuang; Hsieh, Su-Huei; Hsu, John T. -A.; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:09:36Z Design and Structural Analysis of Novel Pharmacophores for Potent and Selective Peroxisome Proliferator-activated Receptor gamma Agonists Lin, Chia-Hui; Peng, Yi-Hui; Coumar, Mohane Selvaraj; Chittimalla, Santhosh Kumar; Liao, Chun-Chen; Lyn, Ping-Chiang; Huang, Chin-Chieh; Lien, Tzu-Wen; Lin, Wen-Hsing; Hsu, John T. -A.; Cheng, Jai-Hong; Chen, Xin; Wu, Jian-Sung; Chao, Yu-Sheng; Lee, Hwei-Jen; Juo, Chiun-Gung; Wu, Su-Ying; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:07:27Z Identification, SAR Studies, and X-ray Co-crystallographic Analysis of a Novel Furanopyrimidine Aurora Kinase A Inhibitor Coumar, Mohane Selvaraj; Tsai, Ming-Tsung; Chu, Chang-Ying; Uang, Biing-Jiun; Lin, Wen-Hsing; Chang, Chun-Yu; Chang, Teng-Yuan; Leou, Jiun-Shyang; Teng, Chi-Huang; Wu, Jian-Sung; Fang, Ming-Yu; Chen, Chun-Hwa; Hsu, John T-A; Wu, Su-Ying; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:07:23Z Anti-Influenza Drug Discovery: Structure-Activity Relationship and Mechanistic Insight into Novel Angelicin Derivatives Yeh, Jiann-Yih; Coumar, Mohane Selvaraj; Horng, Jim-Tong; Shiao, Hui-Yi; Kuo, Fu-Ming; Lee, Hui-Ling; Chen, In-Chun; Chang, Chun-Wei; Tang, Wen-Fang; Tseng, Sung-Nain; Chen, Chi-Jene; Shih, Shin-Ru; Hsu, John T. -A; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立交通大學 2014-12-08T15:06:34Z Fast-Forwarding Hit to Lead: Aurora and Epidermal Growth Factor Receptor Kinase Inhibitor Lead Identification Coumar, Mohane Selvaraj; Chu, Chang-Ying; Lin, Cheng-Wei; Shiao, Hui-Yi; Ho, Yun-Lung; Reddy, Randheer; Lin, Wen-Hsing; Chen, Chun-Hwa; Peng, Yi-Hui; Leou, Jiun-Shyang; Lien, Tzu-Wen; Huang, Chin-Ting; Fang, Ming-Yu; Wu, Szu-Huei; Wu, Jian-Sung; Chittimalla, Santhosh Kumar; Song, Jen-Shin; Hsu, John T. -A.; Wu, Su-Ying; Liao, Chun-Chen; Chao, Yu-Sheng; Hsieh, Hsing-Pang
國立成功大學 2014-09 Aurora kinase inhibitor patents and agents in clinical testing: an update (2011-2013) Cheung, Chun Hei Antonio; Sarvagalla, Sailu; Lee, Jane Ying-Chieh; Huang, Yi-Chun; Coumar, Mohane Selvaraj
國立成功大學 2011-08-24 BPR1K653, a Novel Aurora Kinase Inhibitor, Exhibits Potent Anti-Proliferative Activity in MDR1 (P-gp170)-Mediated Multidrug-Resistant Cancer Cells Cheung, Chun Hei Antonio; Lin, Wen-Hsing; Hsu, John Tsu-An; Hour, Tzyh-Chyuan; Yeh, Teng-Kuang; Ko, Shengkai; Lien, Tzu-Wen; Coumar, Mohane Selvaraj; Liu, Jin-Fen; Lai, Wen-Yang; Shiao, Hui-Yi; Lee, Tian-Ren; Hsieh, Hsing-Pang; Chang, Jang-Yang

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