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教育部委託研究計畫      計畫執行:國立臺灣大學圖書館
 
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機構 日期 題名 作者
國家衛生研究院 2016-10 BPR1J373, an oral multiple tyrosine kinase inhibitor, targets c-KIT for the treatment of c-KIT driven myeloid leukemia Chen, LT;Chen, CT;Jiaang, WT;Chen, TY;Butterfield, JH;Shih, NY;Hsu, JT;Lin, HY;Lin, SF;Tsai, HJ
國家衛生研究院 2016-09 Mycotoxin patulin suppresses innate immune responses by mitochondrial dysfunction and p62/sequestosome-1-dependent mitophagy Tsai, WT;Lo, YC;Wu, MS;Li, CY;Kuo, YP;Lai, YH;Tsai, Y;Chen, KC;Chuang, TH;Yao, CH;Lee, JC;Hsu, LC;Hsu, JT;Yu, GY
國家衛生研究院 2016-02-26 Using mutagenesis to explore conserved residues in the RNA-binding groove of influenza A virus nucleoprotein for antiviral drug development Liu, CL;Hung, HC;Lo, SC;Chiang, CH;Chen, IJ;Hsu, JT;Hou, MH
國家衛生研究院 2016-01-01 Bispecific antibody conjugated manganese-based magnetic engineered iron oxide for imaging of HER2/neu- and EGFR-expressing tumors Wu, SC;Chen, YJ;Wang, HC;Chou, MY;Chang, TY;Yuan, SS;Chen, CY;Hou, MF;Hsu, JT;Wang, YM
國家衛生研究院 2015-10 Identification of substituted naphthotriazolediones as novel tryptophan 2,3-dioxygenase (TDO) inhibitors through structure-based virtual screening Wu, JS;Lin, SY;Liao, FY;Hsiao, WC;Lee, LC;Peng, YH;Hsieh, CL;Wu, MH;Song, JS;Yueh, A;Chen, CH;Yeh, SH;Liu, CY;Lin, SY;Yeh, TK;Hsu, JT;Shih, C;Ueng, SH;Hung, MS;Wu, SY
國家衛生研究院 2015-06-29 Homology modeling of DFG-in FMS-like tyrosine kinase 3 (FLT3) and structure-based virtual screening for inhibitor identification Ke, YY;Singh, VK;Coumar, MS;Hsu, YC;Wang, WC;Song, JS;Chen, CH;Lin, WH;Wu, SH;Hsu, JT;Shih, C;Hsieh, HP
國家衛生研究院 2015-06-16 Anchor-based classification and type-C inhibitors for tyrosine kinases Hsu, KC;Sung, TY;Lin, CT;Chiu, YY;Hsu, JT;Hung, HC;Sun, CM;Barve, I;Chen, WL;Huang, WC;Huang, CT;Chen, CH;Yang, JM
國立交通大學 2014-12-08T15:17:02Z Study of InGaN multiple quantum dots by metal organic chemical vapor deposition Wang, TC; Kuo, HC; Lu, TC; Tsai, CE; Tsai, MY; Hsu, JT; Yang, JR
國家衛生研究院 2014-08 Ligand efficiency based approach for efficient virtual screening of compound libraries Ke, YY;Coumar, MS;Shiao, HY;Wang, WC;Chen, CW;Song, JS;Chen, CH;Lin, WH;Wu, SH;Hsu, JT;Chang, CM;Hsieh, HP
國家衛生研究院 2013-06-28 Optimization of ligand and lipophilic efficiency to identify an in vivo active furano-pyrimidine aurora kinase inhibitor Shiao, HY;Coumar, MS;Chang, CW;Ke, YY;Chi, YH;Chu, CY;Sun, HY;Chen, CH;Lin, WH;Fung, KS;Kuo, PC;Huang, CT;Chang, KY;Lu, CT;Hsu, JT;Chen, CT;Jiaang, WT;Chao, YS;Hsieh, HP
國家衛生研究院 2013-05 Aurora kinase inhibitors reveal mechanisms of HURP in nucleation of centrosomal and kinetochore microtubules Wu, JM;Chen, CT;Coumar, MS;Lin, WH;Chen, ZJ;Hsu, JT;Peng, YH;Shiao, HY;Chu, CY;Wu, JS;Lin, CT;Chen, CP;Hsueh, CC;Chang, KY;Kao, LP;Huang, CY;Chao, YS;Wu, SY;Hsieh, HP;Chi, YH
國家衛生研究院 2013-05 Protein kinase inhibitor design by targeting the Asp-Phe-Gly (DFG) motif: The role of the DFG motif in the design of epidermal growth factor receptor inhibitors Peng, YH;Shiao, HY;Tu, CH;Liu, PM;Hsu, JT;Amancha, PK;Wu, JS;Coumar, MS;Chen, CH;Wang, SY;Lin, WH;Sun, HY;Chao, YS;Lyu, PC;Hsieh, HP;Wu, SY
國家衛生研究院 2013-02-20 Parallel screening of Wild-Type and drug-resistant targets for anti-resistance neuraminidase inhibitors Hsu, KC;Hung, HC;Horng, JT;Fang, MY;Chang, CY;Li, LT;Chen, IJ;Chen, YC;Chou, DL;Chang, CW;Hsieh, HP;Yang, JM;Hsu, JT
國家衛生研究院 2012-09 Anti-influenza drug discovery: Identification of an orally bioavailable quinoline derivative through activity- and property-guided lead optimization Yeh, JY;Coumar, MS;Shiao, HY;Lin, TJ;Lee, YC;Hung, HC;Ko, S;Kuo, FM;Fang, MY;Huang, YL;Hsu, JT;Yeh, TK;Shih, SR;Chao, YS;Horng, JT;Hsieh, HP
國家衛生研究院 2012-08 Development of an anti-influenza drug screening assay targeting nucleoproteins with tryptophan fluorescence quenching Hung, HC;Liu, CL;Hsu, JT;Horng, JT;Fang, MY;Wu, SY;Ueng, SH;Wang, MY;Yaw, CW;Hou, MH
國家衛生研究院 2012-06-07 3-Phenyl-1H-5-pyrazolylamine-based derivatives as potent and efficacious inhibitors of FMS-like tyrosine kinase-3 (FLT3) Hsu, JT;Yeh, TK;Yen, SC;Chen, CT;Hsieh, SY;Hsu, T;Lu, CT;Chen, CH;Chou, LH;Chiu, CH;Chang, YI;Tseng, YJ;Yen, KR;Chao, YS;Lin, WH;Jiaang, WT
國家衛生研究院 2012-06 EGFR and myosin II inhibitors cooperate to suppress EGFR-T790M-mutant NSCLC cells Chiu, HC;Chang, TY;Huang, CT;Chao, YS;Hsu, JT
國家衛生研究院 2012-02 Identification of BPR3P0128 as an Inhibitor of cap-snatching activities of influenza virus Hsu, JT;Yeh, JY;Lin, TJ;Li, ML;Wu, MS;Hsieh, CF;Chou, YC;Tang, WF;Lau, KS;Hung, HC;Fang, MY;Ko, S;Hsieh, HP;Horng, JT
國家衛生研究院 2012-01 BPR1J-097, a novel FLT3 kinase inhibitor, exerts potent inhibitory activity against AML Lin, WH;Jiaang, WT;Chen, CW;Yen, KJ;Hsieh, SY;Yen, SC;Chen, CP;Chang, KY;Chang, CY;Chang, TY;Huang, YL;Yeh, TK;Chao, YS;Chen, CT;Hsu, JT
國家衛生研究院 2012-01 A High-throughput cell-based screening for L858R/T790M mutant epidermal growth factor receptor inhibitors Lin, WH;Song, JS;Lien, TW;Chang, CY;Wu, SH;Huang, YW;Chang, TY;Fang, MY;Yen, KJ;Chen, CH;Chu, CY;Hsieh, HP;Chen, YR;Chao, YS;Hsu, JT
國家衛生研究院 2011-07 Discovery and evaluation of 3-phenyl-1H-5-pyrazolylamine-based derivatives as potent, selective and efficacious inhibitors of FMS-like tyrosine kinase-3 (FLT3) Lin, WH;Hsieh, SY;Yen, SC;Chen, CT;Yeh, TK;Hsu, T;Lu, CT;Chen, CP;Chen, CW;Chou, LH;Huang, YL;Cheng, AH;Chang, YI;Tseng, YJ;Yen, KR;Chao, YS;Hsu, JT;Jiaang, WT
中國醫藥大學 2011-07 Akt pathway is required for oestrogen-mediated attenuation of lung injury in a rodent model of cerulein-induced acute pancreatitis. (Yang SJ); (Chen HM); 謝奇勳(Chi-Hsun Hsieh); (Hsu JT); (Yeh CN); (Yeh TS); (Hwang TL); (Jan YY)*; (Chen MF)
國家衛生研究院 2011-06-01 Suppression of Stat3 activity sensitizes gefitinib-resistant non small cell lung cancer cells Chiu, HC;Chou, DL;Huang, CT;Lin, WH;Lien, TW;Yen, KJ;Hsu, JT
國家衛生研究院 2011-06 Synergistic inhibition of enterovirus 71 replication by interferon and rupintrivir Hung, HC;Wang, HC;Shih, SR;Teng, IF;Tseng, CP;Hsu, JT
國家衛生研究院 2011-04-25 Diosgenin, a plant-derived sapogenin, exhibits antiviral activity in vitro against hepatitis C virus Wang, YJ;Pan, KL;Hsieh, TC;Chang, TY;Lin, WH;Hsu, JT
國家衛生研究院 2010-10-28 Design and synthesis of tetrahydropyridothieno[2,3-d]pyrimidine scaffold based epidermal growth factor receptor (EGFR) kinase inhibitors: the role of side chain chirality and michael acceptor group for maximal potency Wu, CH;Coumar, MS;Chu, CY;Lin, WH;Chen, YR;Chen, CT;Shiao, HY;Rafi, S;Wang, SY;Hsu, H;Chen, CH;Chang, CY;Chang, TY;Lien, TW;Fang, MY;Yeh, KC;Chen, CP;Yeh, TK;Hsieh, SH;Hsu, JT;Liao, CC;Chao, YS;Hsieh, HP
國家衛生研究院 2010-10 Structural basis for the improved potency of peroxisome proliferator-activated receptor (PPAR) agonists Peng, YH;Coumar, MS;Leou, JS;Wu, JS;Shiao, HY;Lin, CH;Lin, WH;Lien, TW;Chen, X;Hsu, JT;Chao, YS;Huang, CF;Lyu, PC;Hsieh, HP;Wu, SY
國家衛生研究院 2010-06-15 Fast-forwarding hit to lead: Aurora and epidermal growth factor receptor kinase inhibitor lead identification Coumar, MS;Chu, CY;Lin, CW;Shiao, HY;Ho, YL;Reddy, R;Lin, WH;Chen, CH;Peng, YH;Leou, JS;Lien, TW;Huang, CT;Fang, MY;Wu, SH;Wu, JS;Chittimalla, SK;Song, JS;Hsu, JT;Wu, SY;Liao, CC;Chao, YS;Hsieh, HP
國家衛生研究院 2010-02-25 Anti-influenza drug discovery: structure-activity relationship and mechanistic insight into novel angelicin derivatives Yeh, JY;Coumar, MS;Horng, JT;Shiao, HY;Kuo, FM;Lee, HL;Chen, IC;Chang, CW;Tang, WF;Tseng, SN;Chen, CJ;Shih, SR;Hsu, JT;Liao, CC;Chao, YS;Hsieh, HP
國家衛生研究院 2010-01 BPR2-D2 targeting viral ribonucleoprotein complex-associated function inhibits oseltamivir-resistant influenza viruses Shih, SR;Horng, JT;Poon, LL;Chen, TC;Yeh, JY;Hsieh, HP;Tseng, SN;Chiang, C;Li, WL;Chao, YS;Hsu, JT
國家衛生研究院 2009-11 Development of NS3/4A protease-based reporter assay suitable for efficiently assessing hepatitis C virus infection Pan, KL;Lee, JC;Sung, HW;Chang, TY;Hsu, JT
中國醫藥大學 2009-08 Mechanism of salutary effects of estrogen on cardiac function following trauma-hemorrhage: Akt-dependent HO-1 up-regulation. (Hsu JT); (Kan WH); (Hsieh CH); (Choudhry MA); (Bland KI); (Chaudry IH)*
國家衛生研究院 2009-07 Novel antiviral agent DTriP-22 targets RNA-dependent RNA polymerase of enterovirus 71 Chen, TC;Chang, HY;Lin, PF;Chern, JH;Hsu, JT;Chang, CY;Shih, SR
國家衛生研究院 2009-04-23 Design and structural analysis of novel pharmacophores for potent and selective peroxisome proliferator-activated receptor gamma agonists Lin, CH;Peng, YH;Coumar, MS;Chittimalla, SK;Liao, CC;Lyn, PC;Huang, CC;Lien, TW;Lin, WH;Hsu, JT;Cheng, JH;Chen, X;Wu, JS;Chao, YS;Lee, HJ;Juo, CG;Wu, SY;Hsieh, HP
國立臺灣大學 2009 Regulation of bacteriocin production in Ruminococcus flavefaciens C94. Wang, WL; Wang, HT; Chen, CY; Liu, JR; Hsu, JT
國家衛生研究院 2008-11 Amantadine as a regulator of internal ribosome entry site Chen, YJ;Zeng, SJ;Hsu, JT;Horng, JT;Yang, HM;Shih, SR;Chu, YT;Wu, TY
國立臺灣大學 2008-07 Anti-HSV activity of digitoxin and its possible mechanisms Su, CT; Hsu, JT; Hsieh, HP; Lin, PH; Chen, TC; Kao, CL; Lee, CN; Chang, SY
臺北醫學大學 2007 Isocostunolide, a sesquiterpene lactone, induces mitochondrial membrane depolarization and caspase-dependent apoptosis in human melanoma cells. 賴基銘; Chen CN; Huang HH; Wu CL; Lin CP; Hsu JT; Hsieh HP; Chuang SE; Lai GM
中國醫藥大學 2005 Effects of splinted prosthesis supported a wide implant or two implants: a three-dimensional finite element analysis Huang, HL; Huang, JS; Ko, CC; Hsu, JT; Chang, CH; Chen, MYC
國家衛生研究院 2004-10 Emergence of mutation clusters in HCV genome during continuous passage of the virus in Sip-L expressing cells Yeh, CT;Lai, HY;Hwang, DJ;Hsu, JT
國立臺灣海洋大學 2004-07 Inhibition of SARS-CoV replication by niclosamide Wu CJ1; Jan JT; Chen CM; Hsieh HP; Hwang DR; Liu HW; Liu CY; Huang HW; Chen SC; Hong CF; Lin RK; Chao YS; Hsu JT
國立臺灣大學 1996-02 The characters and the influential factors of microorganism growth Chen, CY; Hsu, JT

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