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Showing items 1-50 of 56  (2 Page(s) Totally)
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Institution Date Title Author
國家衛生研究院 2025-07-01 Systematic review of natural briaranes in marine organisms (2020-2024): Chemical structures and bioactivities Zheng, LG;Chang, YC;Tsai, YC;Lo, YH;Chi, WC;Zhang, MM;Tsou, LK;Wen, ZH;Hwang, TL;Chen, YY;Sung, PJ
國家衛生研究院 2025-05-16 Marine-derived STING inhibitors, excavatolide B promote wound repair in full-thickness-incision rats Chang, CK;Wu, ZS;Niu, GH;Chou, YY;Tang, SH;Zhang, MM;Sung, CS;Tung, HT;Tsou, LK;Tang, CC;Sung, PJ;Lo, YH;Wen, ZH
國家衛生研究院 2025-05 Identification of PTGR2 inhibitors as a new therapeutic strategy for diabetes and obesity Chang, YC;Hsieh, ML;Lee, HL;Hee, SW;Chang, CF;Yen, HY;Chen, YA;Chen, YR;Chou, YW;Li, FA;Ke, YY;Chen, SY;Hung, MS;Hung, AF;Huang, JY;Chiu, CH;Lin, SY;Shih, SF;Hsu, CN;Hwang, JJ;Yeh, TK;Cheng, TR;Liao, KC;Laio, D;Lin, SW;Chen, TY;Hu, CM;Vogel, U;Saar, D;Kragelund, BB;Tsou, LK;Tseng, YH;Chuang, LM
國家衛生研究院 2025-04-03 Identification of PTGR2 inhibitors as a new therapeutic strategy for diabetes and obesity[Erratum:EMBO Molecular Medicine. 2025 Mar 21;Article in Press.] Chang, YC;Hsieh, ML;Lee, HL;Hee, SW;Chang, CF;Yen, HY;Chen, YA;Chen, YR;Chou, YW;Li, FA;Ke, YY;Chen, SY;Hung, MS;Hung, AF;Huang, JY;Chiu, CH;Lin, SY;Shih, SF;Hsu, CN;Hwang, JJ;Yeh, TK;Cheng, TR;Liao, KC;Laio, D;Lin, SW;Chen, TY;Hu, CM;Vogel, U;Saar, D;Kragelund, BB;Tsou, LK;Tseng, YH;Chuang, LM
國家衛生研究院 2025-04 Junceellolide Q, a new polyacetoxybriarane from the delicate sea whip octocoral Junceella fragilis Goan, YG;Zhang, MM;Tsou, LK;Wen, ZH;Liaw, CC;Lin, YC;Chien, SY;Wu, YJ;Chen, JJ;Do, HN;Jiang, PL;Sung, PJ
國家衛生研究院 2025-02-27 Orally bioavailable and site-selective covalent STING inhibitor derived from a macrocyclic marine diterpenoid Niu, GH;Hsiao, WC;Lee, PH;Zheng, LG;Yang, YS;Huang, WC;Hsieh, CC;Chiu, TY;Wang, JY;Chen, CP;Huang, CL;You, MS;Kuo, YP;Wang, CM;Wen, ZH;Yu, GY;Chen, CT;Chi, YH;Tung, CW;Hsu, SC;Yeh, TK;Sung, PJ;Zhang, MZM;Tsou, LK
國家衛生研究院 2024-05-30 Poly heterocyclic conjugates and their pharmaceutical uses Shih, C;Tsou, LK;Huang, KH;Chen, CT
國家衛生研究院 2024-05-28 Chlorine-containing polyacetoxybriarane diterpenoids from the octocoral Junceella fragilis Do, HN;Chen, YT;Chien, SY;Chen, YY;Zhang, MM;Tsou, LK;Chen, JJ;Wen, ZH;Lo, YH;Zheng, LG;Sung, PJ
國家衛生研究院 2024-03-26 Heterocyclic compounds and use thereof Shia, KS;Chao, YS;Jan, JJ;Tsou, LK;Chen, CT
國家衛生研究院 2024-03 Immunomodulatory and anti-angiogenesis effects of excavatolide B and its derivatives in alleviating atopic dermatitis Chen, HW;Liu, FC;Kuo, HM;Tang, SH;Niu, GH;Zhang, MM;Tsou, LK;Sung, PJ;Wen, ZH
國家衛生研究院 2024-01-23 Poly heterocyclic conjugates and their pharmaceutical uses Tsou, LK;Huang, KH;Chen, CT;Shih, C
國家衛生研究院 2023-12-26 PTGR2 inhibitors and their use Tsou, LK;Hung, MS;Chen, CW;Hsieh, ML;Chang, YC;Chuang, LM
國家衛生研究院 2023-12-19 Heterocyclic compounds and use thereof Chao, YS;Shia, KS;Jan, JJ;Tsou, LK;Chen, CT
國家衛生研究院 2023-10 16-Hydroxybriaranes from the octocoral Briareum stechei Liu, CJ;Wang, CC;Chang, CF;Zhang, MM;Tsou, LK;Wen, ZH;Hwang, TL;Chen, YY;Sung, PJ
國家衛生研究院 2023-09-26 Composto de fórmula (i) e composição farmacêutica Chen, CT;Jan, JJ;Shia, KS;Tsou, LK;Chao, YS
國家衛生研究院 2023-08-31 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2023-08-15 Composto e composição farmacêutica Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2023-07-18 Marine diterpenoid targets STING palmitoylation in mammalian cells Hsiao, WC;Niu, GH;Lo, CF;Wang, JY;Chi, YH;Huang, WC;Tung, CW;Sung, PJ;Tsou, LK;Zhang, MM
國家衛生研究院 2023-05-11 Induction of immune responses and phosphatidylserine exposure by TLR9 activation results in a cooperative antitumor effect with a phosphatidylserine-targeting prodrug Tseng, JC;Yang, JX;Lee, CY;Lo, CF;Liu, YL;Zhang, MM;Huang, LR;Liu, KJ;Wang, CC;Huang, CYF;Hong, YR;Tsou, LK;Chuang, TH
國家衛生研究院 2023-02-13 Briavioid D, a rare 7Beta,8Beta-epoxybriarane from Briareum violaceum Huynh, TH;Ko, CY;Liu, HT;Chen, YP;Zhang, MM;Tsou, LK;Wen, ZH;Chien, SY;Sung, PJ
國家衛生研究院 2023-02-10 Heterocyclic compounds and use thereof Chao, YS;Shia, KS;Jan, JJ;Tsou, LK;Chen, CT
國家衛生研究院 2023-01-10 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2022-09-26 Targeting the phosphatidylserine-immune checkpoint with a small-molecule maytansinoid conjugate Lo, CF;Chiu, TY;Liu, YT;Pan, PY;Liu, KL;Hsu, CY;Fang, MY;Huang, YC;Yeh, TK;Hsu, TA;Chen, CT;Huang, LR;Tsou, LK
國家衛生研究院 2022-07-20 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2022-07 Rejuvenating hepatic tumor microenvironment immunity with a phosphatidylserine-targeting small molecule drug conjugate Huang, KH;Liu, YT;Pan, PY;Lo, CF;Liu, KL;Yeh, TK;Huang, LR;Tsou, LK
國家衛生研究院 2022-06-21 Synthesis and evaluation of small molecule drug conjugates harnessing thioester-linked maytansinoids Lo, CF;Chiu, TY;Liu, YT;Huang, LR;Yeh, TK;Huang, KH;Liu, KL;Hsu, CY;Fang, MY;Huang, YC;Hsu, TA;Chen, CT;Tsou, LK
國家衛生研究院 2022-02-15 Click chemistry and multicomponent reaction for linker diversification of zinc dipicolylamine-based drug conjugates Tsai, CH;Chiu, TY;Chen, CT;Hsu, CY;Tsai, YR;Yeh, TK;Huang, KH;Tsou, LK
國家衛生研究院 2021-10 Chemoproteomic profiling reveals cellular targets of nitro-fatty acids Fang, MY;Huang, KH;Tu, WJ;Chen, YT;Pan, PY;Hsiao, WC;Ke, YY;Tsou, LK;Zhang, MM
國家衛生研究院 2021-03-02 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2021-01-31 Briarenols W-Z: Chlorine-containing polyoxygenated briaranes from octocoral briareum stechei (Kükenthal, 1908) Chen, YY;Zhang, YL;Lee, GH;Tsou, LK;Zhang, MM;Hsieh, HP;Chen, JJ;Ko, CY;Wen, ZH;Sung, PJ
國家衛生研究院 2021-01-05 Derivados de dipicolilamina y sus usos farmacéuticos Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2021-01 BPRDP056, a novel small molecule drug conjugate specifically targeting phosphatidylserine for cancer therapy Chen, YY;Lo, CF;Chiu, TY;Hsu, CY;Yeh, TK;Chen, CP;Huang, CL;Huang, CY;Wang, MH;Huang, YC;Ho, HH;Chao, YS;Shih, JC;Tsou, LK;Chen, CT
中山醫學大學 2021 Chlorinated briarane diterpenoids from octocoral Briareum stechei (Kukenthal, 1908) Huynh, TH; Lee, GH; Tanaka, J; Hsieh, HP; Tsou, LK; Zhang, MZM; Kuo, TJ; Wen, ZH; Lu, CK; Sung, PJ
國家衛生研究院 2020-10-28 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2020-10-08 Comparative study between deep learning and QSAR classifications for TNBC inhibitors and novel GPCR agonist discovery Tsou, LK;Yeh, SH;Ueng, SH;Chang, CP;Song, JS;Wu, MH;Chang, HF;Chen, SR;Shih, C;Chen, CT;Ke, YY
國家衛生研究院 2020-02-13 Heterocyclic compounds and use thereof Chao, YS;Shia, KS;Jan, JJ;Tsou, LK;Chen, CT
國家衛生研究院 2019-10-23 Heterocyclic compounds and use thereof Shia, KS;Jan, JJ;Tsou, LK;Chen, CT;Chao, YS
國家衛生研究院 2019-10-22 A novel flavivirus entry inhibitor, BP34610, discovered through high-throughput screening with dengue reporter viruses Yang, CC;Hu, HS;Lin, HM;Wu, PS;Wu, RH;Tian, JN;Wu, SH;Tsou, LK;Song, JS;Chen, HW;Chern, JH;Chen, CT;Yueh, A
國家衛生研究院 2019-10-17 Dipicolylamine derivatives and pharmaceutical use thereof Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2019-08-28 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2019-07-11 Linker optimization and therapeutic evaluation of phosphatidylserine-targeting zinc dipicolylamine-based drug conjugates Liu, YW;Chen, YY;Hsu, CY;Chiu, TY;Liu, KL;Lo, CF;Fang, MY;Huang, YC;Yeh, TK;Pak, KY;Gray, BD;Hsu, TA;Huang, KH;Shih, C;Shia, KS;Chen, CT;Tsou, LK
國家衛生研究院 2019-07 BPRDP056, a novel small molecule drug conjugate specifically targeting phosphatidylserine for cancer therapy Hsu, CY;Chen, YY;Lo, CF;Chiu, TY;Chen, CP;Huang, CL;Huang, CY;Wang, MH;Chao, YS;Shih, JC;Yeh, TK;Tsou, LK;Chen, CT
國家衛生研究院 2019-05-09 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2019-02-28 Characterization, dynamics, and mechanism of CXCR4 antagonists on a constitutively active mutant Rosenberg, EM, Jr.;Harrison, RES;Tsou, LK;Drucker, N;Humphries, B;Rajasekaran, D;Luker, KE;Wu, CH;Song, JS;Wang, CJ;Murphy, JW;Cheng, YC;Shia, KS;Luker, GD;Morikis, D;Lolis, EJ
國家衛生研究院 2018-03-27 Heterocyclic compounds and use thereof Shia, KS;Jan, JJ;Tsou, LK;Chen, CT;Chao, YS
國家衛生研究院 2018-02-08 Development of stem-cell-mobilizing agents targeting CXCR4 receptor for peripheral blood stem cell transplantation and beyond Wu, CH;Song, JS;Kuan, HH;Wu, SH;Chou, MC;Jan, JJ;Tsou, LK;Ke, YY;Chen, CT;Yeh, KC;Wang, SY;Yeh, TK;Tseng, CT;Huang, CL;Wu, MH;Kuo, PC;Lee, CJ;Shia, KS
國家衛生研究院 2018-01-09 Heterocyclic compounds and use thereof Shia, KS;Jan, JJ;Tsou, LK;Chen, CT;Chao, YS
國家衛生研究院 2017-10-03 Dipicolylamine derivatives and their pharmaceutical uses Chen, CT;Shia, KS;Wu, CH;Tsou, LK;Chao, YS
國家衛生研究院 2017-08-02 Harnessing CXCR4 antagonists in stem cell mobilization, HIV infection, ischemic diseases, and oncology Tsou, LK;Huang, YH;Song, JS;Ke, YY;Huang, JK;Shia, KS
國家衛生研究院 2017-07 Design, synthesis, and evaluation of thiazolidine-2,4-dione derivatives as a novel class of glutaminase inhibitors Yeh, TK;Kuo, CC;Lee, YZ;Ke, YY;Chu, KF;Hsu, HY;Chang, HY;Liu, YW;Song, JS;Yang, CW;Lin, LM;Sun, MW;Wu, SH;Kuo, PC;Shih, C;Chen, CT;Tsou, LK;Lee, SJ

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