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Institution Date Title Author
國家衛生研究院 2014-12 BPR-3P0128 inhibits RNA-dependent RNA polymerase elongation and VPg uridylylation activities of Enterovirus 71 Balaji, VA;Chen, GW;Hsieh, PT;Horng, JT;Hsu, JTA;Hsieh, HP;Chen, TC;Weng, KF;Shih, SR
國家衛生研究院 2013-04-07 BPR000K, a novel Aurora kinase inhibitor Chao, YS;Hsu, JTA;Chen, CT;Yeh, TK;Pan, SL;Hsieh, HP
國家衛生研究院 2011-01 BPR0C261 is a novel orally active antitumor agent with antimitotic and anti-angiogenic activities Hu, CB;Chen, CP;Yeh, TK;Song, JS;Chang, CY;Chuu, JJ;Tung, FF;Ho, PY;Chen, TW;Lin, CH;Wang, MH;Chang, KY;Huang, CL;Lin, HL;Li, WT;Hwang, DR;Chern, JH;Hwang, LL;Chang, JY;Chao, YS;Chen, CT
國家衛生研究院 2022-11-15 BPR0C261, an analogous of microtubule disrupting agent D-24851 enhances the radiosensitivity of human non-small cell lung cancer cells via p53-dependent and p53-independent pathways Leu, JD;Lin, ST;Chen, CT;Chang, CA;Lee, YJ
衛生福利部國家中醫藥研究所 2013 BPR0C305, an orally active microtubule-disrupting anticancer agent Li, Wen-Tai; Yeh, Teng-Kuang; Song, Jen-Shin; Yang, Yung-Ning; Chen, Tung-Wei; Lin, Chi-Hung; Chen, Ching-Ping; Shen, Chien-Chang; Hsieh, Chih-Chien; Lin, Heng-Liang; Chao, Yu-Sheng; Chen, Chiung-Tong
國家衛生研究院 2013-11 BPR0C305, an orally active microtubule-disrupting anticancer agent Li, WT;Yeh, TK;Song, JS;Yang, YN;Chen, TW;Lin, CH;Chen, CP;Shen, CC;Hsieh, CC;Lin, HL;Chao, YS;Chen, CT
國家衛生研究院 2004-07-01 BPR0L075, a novel synthetic indole compound with antimitotic activity in human cancer cells, exerts effective antitumoral activity in vivo Kuo, CC; Hsieh, HP; Pan, WY; Chen, CP; Lion, JP; Lee, SJ; Chang, YL; Chen, LT; Chen, CT; Chang, JY
國家衛生研究院 2012-01 BPR1J-097, a novel FLT3 kinase inhibitor, exerts potent inhibitory activity against AML Lin, WH;Jiaang, WT;Chen, CW;Yen, KJ;Hsieh, SY;Yen, SC;Chen, CP;Chang, KY;Chang, CY;Chang, TY;Huang, YL;Yeh, TK;Chao, YS;Chen, CT;Hsu, JT
國立交通大學 2014-12-08T15:22:05Z BPR1J-097, a novel FLT3 kinase inhibitor, exerts potent inhibitory activity against AML Lin, W-H; Jiaang, W-T; Chen, C-W; Yen, K-J; Hsieh, S-Y; Yen, S-C; Chen, C-P; Chang, K-Y; Chang, C-Y; Chang, T-Y; Huang, Y-L; Yeh, T-K; Chao, Y-S; Chen, C-T; Hsu, J. T-A
國家衛生研究院 2012-11 BPR1J271, a novel FLT3 inhibitor for treating acute myeloid leukemia Chen, CT;Lin, WH;Chou, LH;Chen, CP;Yen, SC;Huang, YL;Yeh, TK;Hsu, JTA;Jiaang, WI;Chao, YS
國家衛生研究院 2018-08-24 BPR1J373, a novel multi-targeted kinase inhibitor, effectively suppresses the growth of gastrointestinal stromal tumor Tsai, HJ;Jiaang, WT;Shih, NY;Fletcher, JA;Lin, MJ;Yang, MY;Chen, CT;Hsu, TJ;Wu, CC;Lin, HY;Chen, LT
國家衛生研究院 2018-08-24 BPR1J373, a novel multitargeted kinase inhibitor, effectively suppresses the growth of gastrointestinal stromal tumor Tsai, HJ;Jiaang, WT;Shih, NY;Fletcher, JA;Lin, MJ;Yang, MY;Chen, CT;Hsu, TAJ;Wu, CC;Lin, HY;Chen, LT
國立成功大學 2018 BPR1J373, a novel multitargeted kinase inhibitor, effectively suppresses the growth of gastrointestinal stromal tumor Tsai, H.-J.;Jiaang, W.-T.;Shih, N.-Y.;Fletcher, J.A.;Lin, M.-J.;Yang, M.-Y.;Chen, Chen C.-T.;Hsu, T.-A.J.;Wu, C.-C.;Lin, H.-Y.;Chen, L.-T.
國家衛生研究院 2016-10 BPR1J373, an oral multiple tyrosine kinase inhibitor, targets c-KIT for the treatment of c-KIT driven myeloid leukemia Chen, LT;Chen, CT;Jiaang, WT;Chen, TY;Butterfield, JH;Shih, NY;Hsu, JT;Lin, HY;Lin, SF;Tsai, HJ
國立成功大學 2016-10-01 BPR1J373, an Oral Multiple Tyrosine Kinase Inhibitor, Targets c-KIT for the Treatment of c-KIT-Driven Myeloid Leukemia Chen, Li-Tzong; Chen, Chiung-Tong; Jiaang, Weir-Torn; Chen, Tsai-Yun; Butterfield, Joseph H.; Shih, Neng-Yao; Hsu, John Tsu-An; Lin, Hui-You; Lin, Sheng-Fung; Tsai, Hui-Jen
國家衛生研究院 2011-08 BPR1K653, a novel aurora kinase inhibitor, exhibits potent anti-proliferative activity in MDR1 (P-gp170)-mediated multidrug-resistant cancer cells Cheung, CH;Lin, WH;Hsu, TA;Hour, TC;Yeh, TK;Ko, S;Lien, TW;Coumar, MS;Liu, JF;Lai, WY;Shiao, HY;Lee, TR;Hsieh, HP;Chang, JY
國立成功大學 2011-08-24 BPR1K653, a Novel Aurora Kinase Inhibitor, Exhibits Potent Anti-Proliferative Activity in MDR1 (P-gp170)-Mediated Multidrug-Resistant Cancer Cells Cheung, Chun Hei Antonio; Lin, Wen-Hsing; Hsu, John Tsu-An; Hour, Tzyh-Chyuan; Yeh, Teng-Kuang; Ko, Shengkai; Lien, Tzu-Wen; Coumar, Mohane Selvaraj; Liu, Jin-Fen; Lai, Wen-Yang; Shiao, Hui-Yi; Lee, Tian-Ren; Hsieh, Hsing-Pang; Chang, Jang-Yang
國家衛生研究院 2011-09-23 BPR1K653, a novel Aurora Kinase Inhibitor, exhibits potent anti-proliferative activity in P-gp170 (MDR1)-mediated VX680-resistant cancer cells in vitro and in vivo Hsieh, HP;Cheung, CHA;Lin, WH;Hsu, TA;Coumar, MS;Chao, YS;Chang, JY
國家衛生研究院 2019-07-03 BPR1M97, a dual mu opioid receptor/nociceptin-orphanin FQ peptide receptor agonist, produces potent antinociceptive effects with safer properties than morphine Chao, PK;Chang, HF;Chang, WT;Yeh, TK;Ou, LC;Chuang, JY;Tsu-An Hsu, J;Tao, PL;Loh, HH;Shih, C;Ueng, SH;Yeh, SH
國立成功大學 2020 BPR1M97, a dual mu opioid receptor/nociceptin-orphanin FQ peptide receptor agonist, produces potent antinociceptive effects with safer properties than morphine Chao, P.-K.;Chang, H.-F.;Chang, W.-T.;Yeh, T.-K.;Ou, L.-C.;Chuang, J.-Y.;Tsu-An, Hsu J.;Tao, P.-L.;Loh, H.H.;Shih, C.;Ueng, S.-H.;Yeh, S.-H.
國家衛生研究院 2010-01 BPR2-D2 targeting viral ribonucleoprotein complex-associated function inhibits oseltamivir-resistant influenza viruses Shih, SR;Horng, JT;Poon, LL;Chen, TC;Yeh, JY;Hsieh, HP;Tseng, SN;Chiang, C;Li, WL;Chao, YS;Hsu, JT
國立交通大學 2014-12-08T15:07:38Z BPR2-D2 targeting viral ribonucleoprotein complex-associated function inhibits oseltamivir-resistant influenza viruses Shih, Shin-Ru; Horng, Jim-Tong; Poon, Leo L. M.; Chen, Tzu-Chun; Yeh, Jiann-Yih; Hsieh, Hsing-Pang; Tseng, Sung-Nain; Chiang, Chiayn; Li, Wan-Ling; Chao, Yu-Sheng; Hsu, John T. -A.
國家衛生研究院 2015-08 BPR2P001S0, a Coumarin derivative, induced cell cycle arrest in A549 through inhibiting PDPK1 activity Lin, PH;Jao, TM;Hung, YL;Hsieh, HP;Yang, YC;Chang, SY
國家衛生研究院 2024-04 BPR3P0128, a non-nucleoside RNA-dependent RNA polymerase inhibitor, inhibits SARS-CoV-2 variants of concern and exerts synergistic antiviral activity in combination with remdesivir Tang, WF;Chang, YH;Lin, CC;Jheng, JR;Hsieh, CF;Chin, YF;Chang, TY;Lee, JC;Liang, PH;Lin, CY;Lin, GH;Cai, JY;Chen, YL;Chen, YS;Tsai, SK;Liu, PC;Yang, CM;Shadbahr, T;Tang, J;Hsu, YL;Huang, CH;Wang, LY;Chen, CC;Kau, JH;Hung, YJ;Lee, HY;Wang, WC;Tsai, HP;Horng, JT
國家衛生研究院 2020-08 BPR6K609: An Aurora kinase inhibitor targeting small cell lung cancer with MYC amplification Chi, YH;Chang, CP;Ke, YY;Lin, WH;Wang, WP;Tsai, CH;Chen, YT;Su, YJ;Hung, MC;Wu, ZW;Wu, MH;Yeh, TK;Chen, CP;Song, JS;Chen, CT;Shih, C

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